BDBM437303 5-(1-Benzyl-1H-pyrazol-4-yl)-4-(3-methanesulfonyl- pyrrolidin-1-yl)-1-methyl-1H-pyridin-2-one::US10617680, Example 37::US11020380, Example 37

SMILES Cn1cc(-c2cnn(Cc3ccccc3)c2)c(cc1=O)N1CCC(C1)S(C)(=O)=O

InChI Key InChIKey=VWKJNTRBWUSUSR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437303   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437303(5-(1-Benzyl-1H-pyrazol-4-yl)-4-(3-methanesulfonyl-...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437303(5-(1-Benzyl-1H-pyrazol-4-yl)-4-(3-methanesulfonyl-...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent