BDBM437658 4-Ethoxy-5-(5-methanesulfonyl-4,5,6,7-tetrahydro- pyrazolo[1,5-a]pyrazin-3-yl)-1-methyl-1H-pyridin-2-one::US10617680, Example 392::US11020380, Example 392

SMILES CCOc1cc(=O)n(C)cc1-c1cnn2CCN(Cc12)S(C)(=O)=O

InChI Key InChIKey=WMVJHZIZWNPUSM-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437658   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437658(4-Ethoxy-5-(5-methanesulfonyl-4,5,6,7-tetrahydro- ...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437658(4-Ethoxy-5-(5-methanesulfonyl-4,5,6,7-tetrahydro- ...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent