BDBM450959 US10676469, Compound 243::US11124504, Cpd. No. 243
SMILES CCc1cc(F)c2nc(N3CC[C@H](C[C@@H]3C)NC3CCOCC3)c(-c3nc(C)no3)c(C)c2c1
InChI Key InChIKey=PHWLVLLLTAYXDP-MGPUTAFESA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 450959
Affinity DataIC50: 55nMAssay Description:The purpose of this assay is to confirm the potency and selectivity of compounds synthesized to be OPRK1 Antagonists. This assay monitors the OPRMu1 ...More data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:The cell line for the OPRK1 antagonist assay stably expresses the following elements: The carboxy terminus of the OPRK1 receptor has a 7-amino acid l...More data for this Ligand-Target Pair