BDBM453277 US10729710, Compound (Ib)
SMILES CCCN1CCC[C@@H]2Cc3c4OCOc4ccc3C[C@@H]12
InChI Key InChIKey=DKFJCEPDDQVHLK-UKRRQHHQSA-N
Data 3 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 453277
Affinity DataEC50: >1.00E+3nMAssay Description:Dopamine D1 receptor agonism was measured using a HTRF cAMP from CisBio using the protocol developed by HD Biosciences (China). Briefly, the assay is...More data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Evaluation of the agonist activity of compounds (I), (Ia) and (Ib) at the human 5-HT2B receptor was performed by Eurofins/Cerep (France) measuring th...More data for this Ligand-Target Pair
Affinity DataEC50: 46nMAssay Description:Dopamine D2 receptor agonism was measured using a calcium mobilization assay protocol developed by HD Biosciences (China). Briefly, HEK293/G15 cells ...More data for this Ligand-Target Pair