BDBM456009 2-(3-(cyclopropylethynyl)-7- (3-methyl-1H-pyrazol-4-yl)- 2H-indazol-2-yl)-N-hydroxy- 3-phenylpropanamide::US10723705, No. I-0166

SMILES Cc1n[nH]cc1-c1cccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO

InChI Key

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 456009   

TargetHistone deacetylase 8(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM456009(2-(3-(cyclopropylethynyl)-7- (3-methyl-1H-pyrazol-...)
Affinity DataIC50: <50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent