BDBM462593 US10766903, Example 205
SMILES OC1(Cn2cnc3n(c(Cl)cc3c2=O)-c2ccc(F)cc2)CCN(CC1)C(=O)c1cnc(o1)C1CC1
InChI Key InChIKey=NELLFLURYUFRHV-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 462593
Affinity DataIC50: <250nMAssay Description:USP7 activity was monitored in a fluorescence polarisation (FP) homogeneous assay using the isopeptide ubiquitin-Lys-TAMRA substrate (U-558, Boston B...More data for this Ligand-Target Pair