BDBM484073 (S)-1-((R)-8-(1H- pyrrolo[3,2-b]pyridin-6- ylsulfonyl)-1-oxa-8- azaspiro[4.5]decan-3- ylamino)-3-(3- (mcthylsulfonyl)phenoxy) propan-2-ol::US10927123, Compound 320::US10927123, Compound 321

SMILES CS(=O)(=O)c1cccc(OC[C@@H](O)CN[C@H]2COC3(C2)CCN(CC3)S(=O)(=O)c2cnc3cc[nH]c3c2)c1

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 484073   

TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM484073((S)-1-((R)-8-(1H- pyrrolo[3,2-b]pyridin-6- ylsulfo...)
Affinity DataIC50:  1.78E+4nMAssay Description:Compounds were dissolved and serially diluted (5-fold) in DMSO to generate a 10-point dose response stock. The stock was then diluted 100-fold in ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM484073((S)-1-((R)-8-(1H- pyrrolo[3,2-b]pyridin-6- ylsulfo...)
Affinity DataIC50:  1.12E+4nMAssay Description:Compounds were dissolved and serially diluted (5-fold) in DMSO to generate a 10-point dose response stock. The stock was then diluted 100-fold in ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent