BDBM492881 N-((5-chloro-1H- indazol-3-yl)methyl)-6- (methyl(4-((2- oxopyridin-1(2H)- yl)methyl)phenyl)amino) picolinamide::US10981893, Example 10

SMILES CN(c1ccc(Cn2ccccc2=O)cc1)c1cncc(c1)C(=O)NCc1n[nH]c2ccc(Cl)cc12

InChI Key InChIKey=HCMPSPCOWLYFIS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 492881   

TargetPlasma kallikrein(Homo sapiens (Human))
Attune Pharmaceuticals

US Patent
LigandPNGBDBM492881(N-((5-chloro-1H- indazol-3-yl)methyl)-6- (methyl(4...)
Affinity DataIC50:  1.00E+4nMAssay Description:The ability of the compounds disclosed herein to inhibit human plasma kallikrein activity was quantified according to the procedures below.A 10 mM so...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent