BDBM495127 US10995084, Ex. No. 4B-33
SMILES C[C@@H](NC(=O)c1ccc(Oc2cc(C)n[nH]c2=O)c(C)n1)C(=O)N1[C@H](CC[C@H]1c1cccc(Cl)c1)[C@H](C)N(CC(F)(F)F)C(C)=O
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 495127
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Kissei Pharmaceutical
US Patent
Kissei Pharmaceutical
US Patent
Affinity DataKi: 0.0500nMAssay Description:The binding affinity assay of compounds for human CGRP receptor was carried out by inhibition of radiolabeled ligand [125I]-CGRP binding in human neu...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Kissei Pharmaceutical
US Patent
Kissei Pharmaceutical
US Patent
Affinity DataIC50: 0.0300nMAssay Description:The binding affinity assay of compounds for human CGRP receptor was carried out by inhibition of radiolabeled ligand [125I]-CGRP binding in human neu...More data for this Ligand-Target Pair