BDBM50000278 2-(3,4-Dichloro-phenyl)-1-(2-piperidin-1-ylmethyl-piperidin-1-yl)-ethanone::2-(3,4-Dichloro-phenyl)-1-(2-piperidin-1-ylmethyl-piperidin-1-yl)-ethanone(HCl)::CHEMBL131328
SMILES Clc1ccc(CC(=O)N2CCCCC2CN2CCCCC2)cc1Cl
InChI Key InChIKey=PZKHOISBMZGAFR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50000278
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Compound was evaluated for its binding affinity against Opioid receptor kappa 1 subtype in guinea pig brain (minus cerebellum)using [3H]-U-69,593 as ...More data for this Ligand-Target Pair
Affinity DataKi: 4.81E+3nMAssay Description:Compound was evaluated for its binding affinity against Opioid receptor mu 1 subtype in guinea pig brain (minus cerebellum) using [3H]-DAGO as radiol...More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Opioid receptor kappa agonist potency was determined in vitro using rabbit vas deferens(LVD) preparationMore data for this Ligand-Target Pair