BDBM50002905 CHEMBL373535
SMILES CC(Oc1ccccc1-c1cccnc1)C1=NCCN1
InChI Key InChIKey=AFWQDDUMQAQVSC-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 14 hits for monomerid = 50002905
Affinity DataKi: 65nMAssay Description:Displacement of [3H]RX821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Displacement of [3H]RX821002 from human adrenergic alpha2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 933nMAssay Description:Displacement of [3H]RX821002 from human adrenergic alpha-2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 933nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist activity at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonist activity at human adrenergic alpha-2A receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
Affinity DataEC50: 589nMAssay Description:Agonist activity at human adrenergic alpha-2A receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human adrenergic alpha-2B receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonistic potency at human adrenergic alpha2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonistic potency at human adrenergic alpha-2A receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonistic potency at human adrenergic alpha-2B receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human adrenergic alpha-2C receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair