BDBM50009685 9-METHYL-9H-PURIN-6-AMINE::9-Methyl-9H-adenine::9-Methyl-9H-purin-6-ylamine::CHEMBL65976
SMILES Cn1cnc2c(N)ncnc12
InChI Key InChIKey=WRXCXOUDSPTXNX-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 15 hits for monomerid = 50009685
Affinity DataKi: 6.90E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.60E+3nMAssay Description:Binding affinity against Adenosine A2A receptor by using [3H]CGS-21680 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+4nMAssay Description:Affinity for the Adenosine A1 receptor in the absence of GTP (A1-GTP) by using [3H]DPCPX as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+4nMAssay Description:Affinity for the Adenosine A1 receptor in the absence of GTP (A1-GTP) by using [3H]DPCPX as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by using [3H]NECA as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Tested for inhibition of rat PC12 adenylate cyclase stimulation by using NECA as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+4nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by using [3H]- PIA as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))
Smith Kline & French Research
Curated by ChEMBL
Smith Kline & French Research
Curated by ChEMBL
Affinity DataKi: 1.11E+5nMAssay Description:Binding affinity (Ki) against human phosphatidylinositol 4-kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.47E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes with GTPMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))
Smith Kline & French Research
Curated by ChEMBL
Smith Kline & French Research
Curated by ChEMBL
Affinity DataIC50: 1.61E+5nMAssay Description:Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding siteMore data for this Ligand-Target Pair
Affinity DataIC50: >3.50E+5nMAssay Description:Inhibition of purified Cdc2 p34/Cyclin B obtained from M phase oocytes of the starfish Marthasterias glacialis (precipitation at the higher concentra...More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes without GTPMore data for this Ligand-Target Pair