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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50009685'
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50009685(9-METHYL-9H-PURIN-6-AMINE | 9-Methyl-9H-adenine | ...)
Affinity DataKi:  6.90E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50009685(9-METHYL-9H-PURIN-6-AMINE | 9-Methyl-9H-adenine | ...)
Affinity DataKi:  8.60E+3nMAssay Description:Binding affinity against Adenosine A2A receptor by using [3H]CGS-21680 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed