BDBM50015749 (1-Ethyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-isopropyl-amine::CHEMBL6958
SMILES CCc1nnc2c(NC(C)C)nc3ccccc3n12
InChI Key InChIKey=PZAYUXVLYKQPMH-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50015749
Affinity DataKi: 240nMAssay Description:Binding affinity towards adenosine A1 receptor using [3H]-N-cyclohexyladenosine in rat whole brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity against Adenosine-2 receptor with [3H]-NECA in rat striatal membranes.More data for this Ligand-Target Pair
TargetDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B/Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C/Phosphodiesterase(Rattus norvegicus)
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Evaluated for Ca++ dependent phosphodiesterase activity.More data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair