BDBM50019194 4-Chloro-N-[1-(4-chloro-benzoyl)-5-(2-fluoro-phenyl)-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-benzamide::CHEMBL70593

SMILES Fc1ccccc1C1=NC(NC(=O)c2ccc(Cl)cc2)C(=O)N(C(=O)c2ccc(Cl)cc2)c2ccccc12

InChI Key InChIKey=FMPRFCINNRGLNV-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50019194   

TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50019194(4-Chloro-N-[1-(4-chloro-benzoyl)-5-(2-fluoro-pheny...)
Affinity DataIC50:  550nMAssay Description:Half-maximal inhibition of [125I]gastrin binding to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50019194(4-Chloro-N-[1-(4-chloro-benzoyl)-5-(2-fluoro-pheny...)
Affinity DataIC50:  3.70E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-8(+) binding to cholecystokinin receptor from guinea pig brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50019194(4-Chloro-N-[1-(4-chloro-benzoyl)-5-(2-fluoro-pheny...)
Affinity DataIC50:  18nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to cholecystokinin A receptor from rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed