BDBM50022758 CHEMBL1204266::CHEMBL308142::Dibutyl-{3-[4-(8-methyl-imidazo[1,2-a]pyridin-2-yl)-phenoxy]-propyl}-amine::N-butyl-N-(3-(4-(8-methylimidazo[1,2-a]pyridin-2-yl)phenoxy)propyl)butan-1-amine

SMILES CCCCN(CCCC)CCCOc1ccc(cc1)-c1cn2cccc(C)c2n1

InChI Key InChIKey=CQWPZSWNLBUMFT-UHFFFAOYSA-N

Data  3 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50022758   

TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50022758(CHEMBL1204266 | CHEMBL308142 | Dibutyl-{3-[4-(8-me...)
Affinity DataKi:  4nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50022758(CHEMBL1204266 | CHEMBL308142 | Dibutyl-{3-[4-(8-me...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity for human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50022758(CHEMBL1204266 | CHEMBL308142 | Dibutyl-{3-[4-(8-me...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity for human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022758(CHEMBL1204266 | CHEMBL308142 | Dibutyl-{3-[4-(8-me...)
Affinity DataIC50:  600nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in Rabbit cardiac muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed