BDBM50035441 4'-[3-Butyl-1-(3-nitro-phenyl)-5-oxo-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-biphenyl-2-sulfonic acid 2-chloro-benzoylamide::CHEMBL293501

SMILES CCCCc1nn(-c2cccc(c2)[N+]([O-])=O)c(=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)c1ccccc1Cl

InChI Key InChIKey=FZBCCWWEILQSAK-UHFFFAOYSA-N

Data  1 KI  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50035441   

TargetType-2 angiotensin II receptor(RAT)
Neogenesis

Curated by ChEMBL
LigandPNGBDBM50035441(4'-[3-Butyl-1-(3-nitro-phenyl)-5-oxo-1,5-dihydro-[...)
Affinity DataKi:  173nMAssay Description:Binding affinity to Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Neogenesis

Curated by ChEMBL
LigandPNGBDBM50035441(4'-[3-Butyl-1-(3-nitro-phenyl)-5-oxo-1,5-dihydro-[...)
Affinity DataIC50:  173nMAssay Description:In vitro binding affinity against angiotensin II (AT2) receptor to competitively block the specific binding of [125I]- [Sar1,Ile8] AII to a rat mid b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035441(4'-[3-Butyl-1-(3-nitro-phenyl)-5-oxo-1,5-dihydro-[...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at AT1 receptor in rabbit aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
Neogenesis

Curated by ChEMBL
LigandPNGBDBM50035441(4'-[3-Butyl-1-(3-nitro-phenyl)-5-oxo-1,5-dihydro-[...)
Affinity DataIC50:  31nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 2 bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035441(4'-[3-Butyl-1-(3-nitro-phenyl)-5-oxo-1,5-dihydro-[...)
Affinity DataIC50:  31nMAssay Description:Tested for in vitro binding affinity against angiotensin I (AT1) receptor to competitively block the specific binding of [125I]- [Sar1,Ile8] AII to a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed