BDBM50035475 CHEMBL3355723
SMILES CC(C)C[C@H](CC(=O)NO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCCNC(=O)c1ccc(F)cc1)C(N)=O
InChI Key InChIKey=CHCWPXOCMTZBSY-VJTSUQJLSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50035475
TargetMatrix metalloproteinase-17(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant ADAM17 using Mca-PLAQAV-Dpa-RSSSR-NH2More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant MMP2 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrateMore data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant MMP9 catalytic domain using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrateMore data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of human recombinant MMP12 catalytic domain Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 fluorogenic substrateMore data for this Ligand-Target Pair