BDBM50038276 (R,S) 7-[(3-Iodo-allyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalen-2-ol::7-[((E)-3-Iodo-allyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalen-2-ol::7-[(3-Iodo-allyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalen-2-ol::CHEMBL110239
SMILES CCCN(C\C=C\I)C1CCc2ccc(O)cc2C1
InChI Key InChIKey=RTMIJLQPWFKAFE-FPYGCLRLSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 11 hits for monomerid = 50038276
Affinity DataKi: 0.990nMAssay Description:Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.More data for this Ligand-Target Pair
Affinity DataKi: 1.85nMAssay Description:Tested for the inhibitory activity against Dopamine D3 receptor in infected Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Tested for inhibition of the binding of [125I]NCQ298 to dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Tested for the inhibitory activity against sigma receptor rat cerebellarMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [125I]trans-8-OH-PIPAT in membrane homogenates of hippocampal tissue ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Tested for the inhibitory activity against 5-hydroxytryptamine 1A receptor in rat hippocampalMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Tested for the inhibitory activity against D2H (high-affinity states) receptor in infected HEK 293 cells.More data for this Ligand-Target Pair
Affinity DataKi: 265nMAssay Description:Tested for inhibition of the binding of [125I]NCQ298 to D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 265nMAssay Description:Tested for the inhibitory activity against Dopamine D2 receptor in infected Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.480nMAssay Description:Binding affinity was tested against dopamine receptor D3 in rat striatal membarane homogenateMore data for this Ligand-Target Pair
Affinity DataKd: 0.130nMAssay Description:Binding affinity was tested against dopamine receptor D3 in the absence of NaClMore data for this Ligand-Target Pair