BDBM50054472 (5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid ((R)-2-hydroxy-1-methyl-ethyl)-amide::(R)-Methanandamide::CHEMBL120526::Methanandamide
SMILES CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)N[C@H](C)CO
InChI Key InChIKey=SQKRUBZPTNJQEM-FQPARAGTSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 19 hits for monomerid = 50054472
Affinity DataKi: 17.9nMAssay Description:Binding affinity towards cannabinoid receptor 1 from rat forebrain membranes in the presence of phenylmethanesulfonylfluoride (PMSF) using 0.8 nM [3H...More data for this Ligand-Target Pair
Affinity DataKi: 17.9nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor of rat cerebellar membranes by liquid scintillation counting in presence of serine protease inhibitor ...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-CP-55,940 from Cannabinoid receptor 1 of rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Tested for binding affinity to Cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity for the cannabinoid receptor in the presence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]CP-55940 as radioligand in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity for the cannabinoid receptor in the absence of phenylmethanesulfonyl fluoride (PMSF) was determined in rat fore brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity towards cannabinoid receptor 1 from rat forebrain membranes in the absence of phenylmethanesulfonylfluoride (PMSF) using 0.8 nM [3H]...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes in presence of FAAH inhibitor PMSF by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain membranes in absence of FAAH inhibitor PMSF by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranes in absence of FAAH inhibitor PMSF by radioligand binding ass...More data for this Ligand-Target Pair
Affinity DataKi: 585nMAssay Description:Binding affinity towards cannabinoid receptor using [3H]SR-141,716A as radioligand in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 815nMAssay Description:Compound was evaluated for its binding affinity for mouse spleen Cannabinoid receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 815nMAssay Description:Binding affinity to mouse spleen CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 868nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 868nMAssay Description:Binding affinity towards Cannabinoid receptor 2 from mouse spleen membranes using 0.8 nM [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranes in absence of FAAH inhibitor PMSF by radioligand binding ass...More data for this Ligand-Target Pair
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Universidad De Talca
Curated by ChEMBL
Universidad De Talca
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human TASK1 expressed in African green monkey COS cells by whole cell patch clamp assayMore data for this Ligand-Target Pair