BDBM50054804 (1S,2R)-2-(1-Amino-ethyl)-1-phenyl-cyclopropanecarboxylic acid diethylamide::CHEMBL330958

SMILES CCN(CC)C(=O)[C@]1(C[C@H]1C(C)N)c1ccccc1

InChI Key InChIKey=JZWQQSJMOZMVFS-OTZYVQGASA-N

Data  4 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50054804   

TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50054804((1S,2R)-2-(1-Amino-ethyl)-1-phenyl-cyclopropanecar...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]-paroxetine binding on serotonin transporter of rat cerebral cortical synaptic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50054804((1S,2R)-2-(1-Amino-ethyl)-1-phenyl-cyclopropanecar...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]-paroxetine binding on serotonin transporter of rat cerebral cortical synaptic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50054804((1S,2R)-2-(1-Amino-ethyl)-1-phenyl-cyclopropanecar...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of Serotonin transporter in cerebral cortical synaptic membrane of rats using [3H]-paroxetineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50054804((1S,2R)-2-(1-Amino-ethyl)-1-phenyl-cyclopropanecar...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of Serotonin transporter in cerebral cortical synaptic membrane of rats using [3H]-paroxetineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50054804((1S,2R)-2-(1-Amino-ethyl)-1-phenyl-cyclopropanecar...)
Affinity DataIC50:  2.30E+3nMAssay Description:Concentration required to inhibit of N-methyl-D-aspartic acid (NMDA) receptor produced by oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed