BDBM50054878 2-{2-[2-{Acetyl-[(E)-(3-phenyl-acryloyl)]-amino}-3-(4-fluoro-phenyl)-propionylamino]-5-guanidino-pentanoylamino}-4-methyl-pentanoic acid (1-carbamoyl-4-guanidino-butyl)-amide::CHEMBL264643
SMILES CC(C)CC(NC(=O)C(CCCNC(N)=N)NC(=O)C(Cc1ccc(F)cc1)N(C(C)=O)C(=O)C=Cc1ccccc1)C(=O)NC(CCCNC(N)=N)C(N)=O
InChI Key InChIKey=QYYWZPHESRMBSY-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50054878
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.13E+3nMAssay Description:Concentration required to inhibit agonist (SFFLRR-NH2, at 3 uM) induced platelet aggregation by 50%More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Antagonistic activity against tritiated agonist (SFFLRR-NH2, at 25 nM) binding to human platelet membranes measured by the GTPase assayMore data for this Ligand-Target Pair