BDBM50062426 5-(4-Chloro-phenyl)-9-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene::CHEMBL107998

SMILES COc1ccc2OC(c3ccc(Cl)cc3)c3c(ccc4NC(C)(C)C=C(C)c34)-c2c1

InChI Key InChIKey=QHPLLVOQIJWVSH-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50062426   

TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062426(5-(4-Chloro-phenyl)-9-methoxy-2,2,4-trimethyl-2,5-...)
Affinity DataKi:  2.40nMAssay Description:The binding affinity measured using baculovirus-expressed hPR-A in sf21 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062426(5-(4-Chloro-phenyl)-9-methoxy-2,2,4-trimethyl-2,5-...)
Affinity DataEC50:  3.10nMAssay Description:Agonistic activity was measured for modulation of hPR-B (human progesterone receptor) in co-transfected CV-1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed