BDBM50062432 5-(3-Chloro-phenyl)-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene::CHEMBL416411
SMILES CC1=CC(C)(C)Nc2ccc3-c4cc(F)ccc4OC(c4cccc(Cl)c4)c3c12
InChI Key InChIKey=OHLMRBMVXRKABN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50062432
Affinity DataKi: 0.320nMAssay Description:The binding affinity measured using baculovirus-expressed hPR-A in sf21 cells.More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Compound was evaluated for its binding affinity against baculovirus expressed Progesterone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity for human progesterone receptor isoform A expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity for human progesterone receptor isoform A expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 133nMAssay Description:Binding affinity for human glucocorticoid receptor expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Compound was tested for agonistic activity by cotransfection assay against human Progesterone receptor in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Agonistic activity was measured for modulation of hPR-B (human progesterone receptor) in co-transfected CV-1 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Agonistic activity by cotransfection assay against human Progesterone receptor in T47D cellsMore data for this Ligand-Target Pair