BDBM50072709 9-Fluoro-2,2,4,5-tetramethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene::CHEMBL116007
SMILES CC1Oc2ccc(F)cc2-c2ccc3NC(C)(C)C=C(C)c3c12
InChI Key InChIKey=UAXYYPCBGHLJKQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50072709
Affinity DataKi: 1.10nMAssay Description:Binding affinity was determined against hPR-A (human progesterone receptor) using progesterone radioligand in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 456nMAssay Description:Displacement of DHT from human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 749nMAssay Description:Displacement of Dexamethasone from human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity against hPR (human progesterone receptor) compared to that of progesterone (100%)More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity was determined against hPR (human progesterone receptor) compared to that of progesterone (100%)More data for this Ligand-Target Pair