BDBM50076791 CHEMBL10990::Lithium; (S)-4-methylsulfanyl-2-{[2'-methyl-5-(5-p-tolyl-furan-2-ylmethoxymethyl)-biphenyl-2-carbonyl]-amino}-butyrate

SMILES CSCC[C@H](NC(=O)c1ccc(COCc2ccc(o2)-c2ccc(C)cc2)cc1-c1ccccc1C)C([O-])=O

InChI Key InChIKey=KPLVUGOBZAXWSW-LJAQVGFWSA-M

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50076791   

LigandPNGBDBM50076791(CHEMBL10990 | Lithium; (S)-4-methylsulfanyl-2-{[2'...)
Affinity DataEC50:  1.80nMAssay Description:EC50 is measured as inhibition of ras processing in a whole cell assay for farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50076791(CHEMBL10990 | Lithium; (S)-4-methylsulfanyl-2-{[2'...)
Affinity DataIC50:  2.90nMAssay Description:In vitro inhibitory activity of the compound was evaluated against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed