BDBM50077878 CHEMBL3417043::US9611229, 3
SMILES Clc1ccc(c(Cl)c1)-n1cc(NCCN2CCCCC2)nn1
InChI Key InChIKey=LZDOBGCHNLXCAW-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50077878
Affinity DataKi: 31nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in HEK293 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Laboratorios Del Dr. Esteve
US Patent
Laboratorios Del Dr. Esteve
US Patent
Affinity DataKi: 31.1nMAssay Description:Brain membrane preparation and binding assays for the 61-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y. For...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Esteve
Curated by ChEMBL
Esteve
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells at -80 mV holding potential by whole cell patch clamp assayMore data for this Ligand-Target Pair