BDBM50089255 CHEMBL3577906

SMILES C[C@@H](N(Cc1cccc(c1)C(O)=O)C(=O)c1cc2ccccn2n1)c1ccc(F)cc1F

InChI Key InChIKey=HZFSAMSNWXIPCA-OAHLLOKOSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50089255   

TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50089255(CHEMBL3577906)Copy SMILESCopy InChI

Affinity DataIC50:  234nMAssay Description:Antagonist activity against human recombinant TRPM8 expressed in CHO T-rex cells assessed as inhibition of WS12-induced calcium response pre-incubate...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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