BDBM50089259 CHEMBL3577902

SMILES C[C@@H](N(Cc1cccc(c1)C(O)=O)C(=O)c1cnc2ccccc2c1)c1cccc(Cl)c1

InChI Key InChIKey=JRPBUWRZMBYEIQ-QGZVFWFLSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50089259   

TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50089259(CHEMBL3577902)Copy SMILESCopy InChI

Affinity DataIC50:  62nMAssay Description:Antagonist activity against human recombinant TRPM8 expressed in CHO T-rex cells assessed as inhibition of WS12-induced calcium response pre-incubate...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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