BDBM50089260 CHEMBL3577901

SMILES COc1ccc(cc1)C(C)N(Cc1cccc(c1)C(O)=O)C(=O)c1cnc2ccccc2c1

InChI Key InChIKey=CISIDUHYOJBXAM-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50089260   

TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50089260(CHEMBL3577901)Copy SMILESCopy InChI

Affinity DataIC50:  6.10E+3nMAssay Description:Antagonist activity against human recombinant TRPM8 expressed in CHO T-rex cells assessed as inhibition of WS12-induced calcium response pre-incubate...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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