BDBM50091386 1-{4-[3-(1H-Imidazol-4-yl)-propoxy]-phenyl}-ethanone::CHEMBL114129::CHEMBL128851
SMILES CC(=O)c1ccc(OCCCc2cnc[nH]2)cc1
InChI Key InChIKey=FDJSGXRROVCWFT-UHFFFAOYSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50091386
Affinity DataKi: 0.800nMAssay Description:Histamine H3 receptor antagonist activity in an assay with K+ evoked depolarization-induced release of [3H]-histamine from rat synaptosomes.More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Effect on histamine H3 receptors in vitro, on synaptosomes of rat cerebral cortex for the release of [3H]histamineMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibition of [125I]-iodoproxyfan from rat histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Inhibition of [125I]-iodoproxyfan binding to human histamine H3 receptor of CHO-K1 cellsMore data for this Ligand-Target Pair