BDBM50092077 CHEMBL3582414::US9296728, 8
SMILES OC(=O)C(=C\c1ccc(cc1)N(CC#C)CC#C)\C#N
InChI Key InChIKey=YOJPLQRGAYWLBC-SDNWHVSQSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50092077
Affinity DataIC50: 400nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair