BDBM50099902 4-[4-(3-Hydroxy-phenyl)-thiazol-2-yl]-5-methylsulfanyl-thiophene-2-carboxamidine::CHEMBL28849
SMILES CSc1sc(cc1-c1nc(cs1)-c1cccc(O)c1)C(N)=N
InChI Key InChIKey=KLVFDMVKNCAXRG-UHFFFAOYSA-N
Data 6 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50099902
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
3-Dimensional Pharmaceuticals
Curated by ChEMBL
3-Dimensional Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Inhibitory activity against serine protease urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Inhibitory activity of the compound against TrypsinMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
3-Dimensional Pharmaceuticals
Curated by ChEMBL
3-Dimensional Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibitory activity of the compound against tissue plasminogen activatorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+4nMAssay Description:Inhibitory activity of the compound against Thrombin (no observable inhibition at this screening concentration)More data for this Ligand-Target Pair
Affinity DataKi: >3.10E+4nMAssay Description:Inhibitory activity of the compound against Serine protease chymotrypsin (no observable inhibition at this screening concentration)More data for this Ligand-Target Pair
Affinity DataKi: 3.21E+4nMAssay Description:Inhibitory activity of the compound against plasminMore data for this Ligand-Target Pair