BDBM50100745 CHEMBL436887::Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRIF::Des-AA1,2,5-[IAmp9,Tyr11]-SRIF

SMILES CC(C)NCc1ccc(C[C@@H]2NC(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@@H](Cc3ccccc3)NC(=O)[C@@H](CCCCN)NC(=O)[C@H](N)CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@H](NC2=O)[C@@H](C)O)[C@@H](C)O)C(O)=O)cc1

InChI Key InChIKey=FJRAPOZDHJLSPN-KVMFXWMESA-N

Data  10 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50100745   

TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50: >1.00E+3nMAssay Description:Tested for ability to bind to 20 microM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) recept...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for ability to bind to 20 microM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) recept...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50: >1.00E+3nMAssay Description:Tested for ability to bind to 20 microM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) recept...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for ability to bind to 20 microM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) recept...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50:  384nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [Leu8,D-Trp22,125I-Tyr25]SRIF-28 binding to human somatostatin receptor type 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100745(CHEMBL436887 | Des-AA1,2,5-[DTrp8,IAmp9,Tyr11]-SRI...)
Affinity DataIC50:  17.1nMAssay Description:Tested for ability to bind to 20 microM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) recept...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed