BDBM50102453 Ac-D-Nal-[D-(pCl)Phe]-D-Pal-Ser-[Aph(Hor)]-D-[Amf(MeCbm)]-Leu-ILys-Pro-DAla-NH2::CHEMBL414249
SMILES CNC(=O)NCc1ccc(C[C@@H](NC(=O)[C@H](Cc2ccc(NC(=O)[C@H]3CC(=O)NC(=O)N3)cc2)NC(=O)[C@H](CO)NC(=O)[C@@H](Cc2cccnc2)NC(=O)[C@@H](Cc2ccc(Cl)cc2)NC(=O)[C@@H](Cc2ccc3ccccc3c2)NC(C)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCNC(C)C)C(=O)N2CCC[C@H]2C(=O)N[C@H](C)C(N)=O)cc1
InChI Key InChIKey=QGLSXLHKCPEGQC-NMLZNVJISA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50102453
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataKd: 0.794nMAssay Description:Competitive antagonism of GnRH-induced response in the reporter gene assayMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Ferring Research Institute
Curated by ChEMBL
Ferring Research Institute
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Antagonism of human GnHR receptor, determined in a reporter gene assay in HEK293 cellsMore data for this Ligand-Target Pair