BDBM50104987 CHEMBL367445::sodium salt of 4-tert-Butyl-N-{6-[2-(5-thiophen-2-yl-pyrimidin-2-yloxy)-ethoxy]-5-p-tolyl-pyrimidin-4-yl}-benzenesulfonamide
SMILES Cc1ccc(cc1)-c1c([N-]S(=O)(=O)c2ccc(cc2)C(C)(C)C)ncnc1OCCOc1ncc(cn1)-c1cccs1
InChI Key InChIKey=OIXCWSXEMAVSIY-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50104987
Affinity DataIC50: 0.25nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:In vitro for specific binding of [125I]-ET-1 to GHcell expressed in Endothelin B receptorMore data for this Ligand-Target Pair