BDBM50121205 CHEBI:18295::Histamine
SMILES NCCc1c[nH]cn1
InChI Key InChIKey=NTYJJOPFIAHURM-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50121205
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in SK-N-MC cells incubated for 40 min by liquid scintillation...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]NAMH from human H3R expressed in HEK293T cells incubated for 2 hrs by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Agonist activity at human H3R expressed on HEK293T cells assessed as inhibition of forskolin-induced CRE-driven luciferase activity co-incubated with...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at human H3R expressed on SK-N-MC cells assessed as inhibition of forskolin-induced beta galactosidase activity preincubated with fo...More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Agonist activity at human H3R expressed on HEK293T cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair