BDBM50126554 CHEMBL23405::N-{4-[4-(5-Chloro-thiophene-2-carbonyl)-piperazin-1-yl]-phenyl}-N-[3-(4-cyano-benzyl)-3H-imidazol-4-ylmethyl]-benzenesulfonamide

SMILES Clc1ccc(s1)C(=O)N1CCN(CC1)c1ccc(cc1)N(Cc1cncn1Cc1ccc(cc1)C#N)S(=O)(=O)c1ccccc1

InChI Key InChIKey=YAXJDRSJHWDRKG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50126554   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50126554(CHEMBL23405 | N-{4-[4-(5-Chloro-thiophene-2-carbon...)
Affinity DataIC50:  2nMAssay Description:Inhibit of purified bovine Farnesyl protein transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed