BDBM50126557 CHEMBL284508::N-{4-[4-(5-Chloro-thiophene-2-carbonyl)-piperazin-1-yl]-phenyl}-N-(3H-imidazol-4-ylmethyl)-benzenesulfonamide

SMILES Clc1ccc(s1)C(=O)N1CCN(CC1)c1ccc(cc1)N(Cc1cnc[nH]1)S(=O)(=O)c1ccccc1

InChI Key InChIKey=DLJAGEPCQCBENN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50126557   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50126557(CHEMBL284508 | N-{4-[4-(5-Chloro-thiophene-2-carbo...)
Affinity DataIC50:  600nMAssay Description:Inhibit of purified bovine Farnesyl protein transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed