BDBM50130535 CHEMBL3632695
SMILES OC(=O)\C=C\C(O)=O.COc1cc(ccc1COCC(O)CN1CCC(CC1)N1Cc2ccccc2C1=O)C(F)(F)F
InChI Key InChIKey=BAQUUINKTMAUEY-WLHGVMLRSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50130535
TargetSodium channel protein type 1 subunit alpha(Homo sapiens (Human))
Daiichi Sankyo
Curated by ChEMBL
Daiichi Sankyo
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human NaV1.1 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Daiichi Sankyo
Curated by ChEMBL
Daiichi Sankyo
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human NaV1.7 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 1 subunit alpha [1489-1708](Mus musculus)
Daiichi Sankyo
Curated by ChEMBL
Daiichi Sankyo
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of mouse NaV1.1 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Inhibition of mouse NaV1.7 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Daiichi Sankyo
Curated by ChEMBL
Daiichi Sankyo
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human NaV1.5 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair