BDBM50136425 5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyridin-2-ylmethyl-1,2,3,4-tetrahydro-quinolin-3-yl)-amide::CHEMBL136812

SMILES Clc1ccc2[nH]c(cc2c1)C(=O)NC1Cc2ccccc2N(Cc2ccccn2)C1=O

InChI Key InChIKey=RWBPBDNBISBDEB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50136425   

TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136425(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyri...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136425(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyri...)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed