BDBM50145689 CHEMBL80844::[1-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-hydroxy-propionylamino)-propionylamino]-2-(4-guanidino-phenyl)-ethyl]-phosphonic acid diphenyl ester::diphenyl 1-[(N-benzoyloxycarbonyl-D-seryl)-L-alanyl]amino-2-(4-guanidinophenyl)ethanephosphonate
SMILES [#6]-[#6@H](-[#7]-[#6](=O)-[#6@@H](-[#6]-[#8])-[#7]-[#6](=O)-[#8]-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6](-[#6]-c1ccc(cc1)\[#7]=[#6](/[#7])-[#7])P(=O)([#8]-c1ccccc1)[#8]-c1ccccc1
InChI Key InChIKey=GYFYCGMUNLSJCM-XPKRSZDKSA-N
Data 9 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50145689
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp
Curated by ChEMBL
University Of Antwerp
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibitory activity of the compound was tested against Urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory activity of the compound was tested against Tissue type plasminogen activatorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity of the compound was tested against thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibitory activity of the compound was tested against Coagulation factor XaMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp
Curated by ChEMBL
University Of Antwerp
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibitory activity of the compound was tested against plasminMore data for this Ligand-Target Pair