BDBM50149902 CHEMBL3771372

SMILES CCN(C1CCOCC1)c1cc(Cl)cc(C(=O)NCc2c(CC)cc(C)[nH]c2=O)c1C

InChI Key InChIKey=QJVOGWFUQFOCCE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50149902   

TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50149902(CHEMBL3771372)
Affinity DataIC50:  10nMAssay Description:Inhibition of methyltransferase activity of human EZH2 using chicken oligonucleotide as substrate by pull down assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed