BDBM501504 3-methyl-1-[1-methylpropyll-N-[(1-methyl- 1,2,4-triazol-3-yl)methyl]-5-(2-propoxy-3- pyridyl)pyrazolo[4,3-b]pyridin-7-amine, enantiomer 2::US11026923, Example 134

SMILES CCCOc1ncccc1-c1cc(NCc2ncn(C)n2)c(NC(C)CC)c(n1)C(C)=N

InChI Key InChIKey=XJUDCWZJLDFIBG-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 501504   

LigandPNGBDBM501504(3-methyl-1-[1-methylpropyll-N-[(1-methyl- 1,2,4-tr...)
Affinity DataIC50:  0.960nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays was performed in 60 uL samples containing a fixed amount of the PDE1 enzyme (suff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM501504(3-methyl-1-[1-methylpropyll-N-[(1-methyl- 1,2,4-tr...)
Affinity DataIC50:  1.5nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays was performed in 60 uL samples containing a fixed amount of the PDE1 enzyme (suff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM501504(3-methyl-1-[1-methylpropyll-N-[(1-methyl- 1,2,4-tr...)
Affinity DataIC50:  0.120nMAssay Description:PDE1A, PDE1B and PDE1C assays were performed as follows: the assays was performed in 60 uL samples containing a fixed amount of the PDE1 enzyme (suff...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent