BDBM50150823 CHEMBL1365878

SMILES COc1cc2n(C)c(=O)n(C)c2cc1NS(=O)(=O)c1cccc(c1)C#N

InChI Key InChIKey=STNHMRPSFGWNKM-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50150823   

TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50150823(CHEMBL1365878)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed