BDBM50153261 2-[4-(4-Bromo-2-cyano-phenyl)-piperazin-1-yl]-N-(2,4,6-tribromo-3-methyl-phenyl)-acetamide::CHEMBL183466

SMILES Cc1c(Br)cc(Br)c(NC(=O)CN2CCN(CC2)c2ccc(Br)cc2C#N)c1Br

InChI Key InChIKey=YAGRRKYCTXMYMI-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50153261   

TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50153261(2-[4-(4-Bromo-2-cyano-phenyl)-piperazin-1-yl]-N-(2...)
Affinity DataKi:  114nMAssay Description:In vitro ability to inhibit [3H]-6b binding to human Dopamine receptor D4.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50153261(2-[4-(4-Bromo-2-cyano-phenyl)-piperazin-1-yl]-N-(2...)
Affinity DataKi:  936nMAssay Description:In vitro ability to inhibit [3H]-spiperone binding to human Dopamine receptor D4.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50153261(2-[4-(4-Bromo-2-cyano-phenyl)-piperazin-1-yl]-N-(2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity was calculated in calcium flux assay using HEK-293 cells co-transfected with human Dopamine receptor D4.4 and Galphaqo5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed