BDBM50153937 4-Methyl-thiophene-2-carboxylic acid N''-(2-{4-[3-hydroxy-3-(3-hydroxy-phenyl)-3-phenyl-propyl]-[1,4]diazepan-1-yl}-acetyl)-hydrazide::CHEMBL365853

SMILES Cc1csc(c1)C(=O)NNC(=O)CN1CCCN(CCC(O)(c2ccccc2)c2cccc(O)c2)CC1

InChI Key InChIKey=LAXQWBGYKRJGLA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50153937   

TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Institute For Bio-Medical Research

Curated by ChEMBL
LigandPNGBDBM50153937(4-Methyl-thiophene-2-carboxylic acid N''-(2-{4-[3-...)
Affinity DataIC50:  6.40E+3nMAssay Description:Concentration required to inhibit [125I]-MCP-1 (Monocyte Chemoattractant Protein-1) binding to THP-1 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed