BDBM50154291 CHEMBL3775181

SMILES CS(O)(=O)=O.Cc1oc2c(O)c3C(=O)c4ccccc4C(=O)c3c(O)c2c1C(=O)N1CC[C@H](N)C1

InChI Key InChIKey=DKTINRPQDJMJSR-PPHPATTJSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50154291   

TargetAurora kinase B(Homo sapiens (Human))
Mendeleyev University Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of full length human N-terminal GST-HIS6-tagged Aurora B expressed in sf9 cells by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase C(Homo sapiens (Human))
Mendeleyev University Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of full length human N-terminal GST-HIS6-tagged Aurora C expressed in sf9 cells by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
Mendeleyev University Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of human MAP3K7 by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
Mendeleyev University Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of human N-terminal FLAG, C-terminal HIS8-tagged TLK1 expressed in sf9 cells by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Mendeleyev University Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of full length human N-terminal GST-HIS6-tagged PIM1 expressed in sf9 cells by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Mendeleyev University Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of full length human N-terminal GST-HIS6-tagged PIM3 expressed in sf9 cells by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual serine/threonine and tyrosine protein kinase(Homo sapiens (Human))
Mendeleyev University Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of human RIPK5 by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Mendeleyev University Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of human MKNK1 by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed