BDBM50155166 4-(6-Chloro-pyridazin-3-yl)-piperazine-1-carboxylic acid (4-isopropyl-phenyl)-amide::CHEMBL363699
SMILES CC(C)c1ccc(NC(=O)N2CCN(CC2)c2ccc(Cl)nn2)cc1
InChI Key InChIKey=XSKDODVTPLNVBZ-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50155166
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma
Curated by ChEMBL
Purdue Pharma
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair
TargetPantothenate kinase 3(Homo sapiens (Human))
St. Jude Children'S Research Hospital
Curated by ChEMBL
St. Jude Children'S Research Hospital
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human recombinant N-terminal His6-fusion tagged PanK3 expressed in Escherichia coli BL21 (DE3) measured after 10 mins in presence of AT...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Purdue Pharma
Curated by ChEMBL
Purdue Pharma
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair