BDBM50155969 2-[8-(Butyl-ethyl-amino)-6-methyl-2-oxo-2,3-dihydro-1H-pyrido[2,3-b]pyrazin-4-yl]-5-chloro-benzonitrile; TFA::CHEMBL433592

SMILES CCCCN(CC)c1cc(C)nc2N(CC(=O)Nc12)c1ccc(Cl)cc1C#N

InChI Key InChIKey=RHQHGBKBTVUTBS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50155969   

TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50155969(2-[8-(Butyl-ethyl-amino)-6-methyl-2-oxo-2,3-dihydr...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [125I]-ovine-CRF binding to corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed